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neuropeptide FF

功能和特点
有货

库存信息

关闭

库存信息

关闭
货号 (SKU) 包装规格 是否现货 价格 数量
rp174614-500μg
500μg 期货 Stock Image
rp174614-1mg
1mg 期货 Stock Image

基本描述

产品名称 neuropeptide FF

产品规格参数

CAS编号和信息 rp174614

靶标

Target ID 150
名称 MAS1
缩写名 SHP2
家族 Class A Orphans
别名 m3
基因和蛋白信息
Species Transmembrane Domains Amino Acids Chromosomal Location Gene Symbol Gene Name
Rat 7 324 1q11 Mas1 MAS1 proto-oncogene, G protein-coupled receptor
Human 7 325 6q25.3 MAS1 MAS1 proto-oncogene, G protein-coupled receptor
Mouse 7 324 17 8.69 cM Mas1 MAS1 oncogene
RefSeq Protein NP_036889 (Rn) , NP_002368 (Hs) , NP_032578 (Mm)
UniProtKB P12526 (Rn) , P04201 (Hs) , P30554 (Mm)
OMIM 165180 (Hs)
RefSeq Nucleotide NM_002377 (Hs) , NM_012757 (Rn) , NM_008552 (Mm)
Entrez Gene 4142 (Hs) , 25153 (Rn) , 17171 (Mm)
Ensembl Gene ENSG00000130368 (Hs) , ENSMUSG00000068037 (Mm) , ENSRNOG00000014971 (Rn)
Protein GI 31543241 (Mm) , 4505105 (Hs) , 6981186 (Rn)
GPCRdb mas_human (Hs) , mas_mouse (Mm) , mas_rat (Rn)
UniProtKB ID/Entry name MAS_HUMAN (Hs) , MAS_MOUSE (Mm) , MAS_RAT (Rn)
ChEMBL Target CHEMBL3559701 (Hs)
Target ID 300
名称 NPFF1 receptor
缩写名 SHP2
家族 Neuropeptide FF/neuropeptide AF receptors
别名 AII β
基因和蛋白信息
Species Transmembrane Domains Amino Acids Chromosomal Location Gene Symbol Gene Name
Rat 7 432 20q11 Npffr1 neuropeptide FF receptor 1
Human 7 430 10q22.1 NPFFR1 neuropeptide FF receptor 1
Mouse 7 432 10 32.24 cM Npffr1 neuropeptide FF receptor 1
RefSeq Protein NP_071627 (Rn) , NP_071429 (Hs) , NP_001170982 (Mm)
UniProtKB Q9EP86 (Rn) , Q9GZQ6 (Hs)
OMIM 607448 (Hs)
RefSeq Nucleotide NM_022146 (Hs) , NM_022291 (Rn) , NM_001177511 (Mm)
Entrez Gene 64106 (Hs) , 64107 (Rn) , 237362 (Mm)
Ensembl Gene ENSG00000148734 (Hs) , ENSMUSG00000020090 (Mm) , ENSRNOG00000000559 (Rn)
Protein GI 11545887 (Hs) , 294661831 (Rn) , 294661833 (Mm)
GPCRdb npff1_human (Hs) , npff1_rat (Rn)
UniProtKB ID/Entry name NPFF1_HUMAN (Hs) , NPFF1_RAT (Rn)
ChEMBL Target CHEMBL4571 (Rn) , CHEMBL5951 (Hs)
Target ID 301
名称 NPFF2 receptor
缩写名 SHP2
家族 Neuropeptide FF/neuropeptide AF receptors
别名 AII β
基因和蛋白信息
Species Transmembrane Domains Amino Acids Chromosomal Location Gene Symbol Gene Name
Rat 7 417 14p22 Npffr2 neuropeptide FF receptor 2
Human 7 522 4q13.3 NPFFR2 neuropeptide FF receptor 2
Mouse 7 417 5 E1 Npffr2 neuropeptide FF receptor 2
RefSeq Protein NP_076470 (Rn) , NP_573455 (Mm) , NP_444264 (Hs) , NP_001138228 (Hs) , NP_004876 (Hs)
UniProtKB Q9EQD2 (Rn) , Q924H0 (Mm) , Q9Y5X5 (Hs)
OMIM 607449 (Hs)
RefSeq Nucleotide NM_023980 (Rn) , NM_133192 (Mm) , NM_001144756 (Hs) , NM_004885 (Hs) , NM_053036 (Hs)
Entrez Gene 10886 (Hs) , 78964 (Rn) , 104443 (Mm)
Ensembl Gene ENSG00000056291 (Hs) , ENSMUSG00000035528 (Mm) , ENSRNOG00000003067 (Rn)
Protein GI 13027438 (Rn) , 221316654 (Hs) , 31981539 (Mm)
GPCRdb npff2_human (Hs) , npff2_mouse (Mm) , npff2_rat (Rn)
UniProtKB ID/Entry name NPFF2_HUMAN (Hs) , NPFF2_MOUSE (Mm) , NPFF2_RAT (Rn)
ChEMBL Target CHEMBL4523416 (Mm) , CHEMBL3425 (Rn) , CHEMBL5952 (Hs)

关联配体

Ligand ID 1479
名称 neuropeptide FF
类别 Peptide
学名 4-amino-N-(4,6-dimethylpyrimidin-2-yl)benzenesulfonamide
生物活性评价 The sulfonamide class of antibacterial compounds are primarily bacteriostatic agents and have a broad spectrum of activity against both Gram-positive and Gram-negative species of bacteria (reviewed in ).
评价 Sulfadimidine (sulfamethazine) is a sulfonamide antibacterial compound. This class of compounds are competitive inhibitors of bacterial dihydropteroate synthase (DHPS), an enzyme in the pathway which generates the folic acid that is essential for bacterial growth.
配体家族 Neuropeptides
基因/前体
Gene symbol Gene name Precursor protein name Species 别名
Npff neuropeptide FF-amide peptide precursor neuropeptide FF-amide peptide precursor Rat FMRFamide-related peptides, neuropeptide FF-amide peptide precursor
NPFF neuropeptide FF-amide peptide precursor neuropeptide FF-amide peptide precursor Human FMRFAL
单字母多肽序列 FLFQPQRF
三字母多肽序列 Phe-Leu-Phe-Gln-Pro-Gln-Arg-Phe-NH2
翻译后修饰 Amidation of C-terminal phenylalanine
化学修饰

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