| 货号 (SKU) | 包装规格 | 是否现货 | 价格 | 数量 |
|---|---|---|---|---|
| Lib412031-100μl-well | 100μl/well |
期货  |
| |
| Lib412031-2×100μl-well | 2×100μl/well |
期货 |
|
| 英文名称 | GPCR Compound Library |
|---|---|
| 储存温度 | -80℃储存 |
| 运输条件 | 超低温冰袋运输 |
| 产品介绍 |
描述及优势 ? 提供1325种靶向G蛋白偶联受体的小分子，可用于高通量筛选和高内涵筛选 ? GPCR化合物库中的所有小分子都具有良好的生物和药学活性 ? 一项发现GPCR药物是最丰富信号受体的有力工具 ? 据估计大约200个“孤儿”GPCR功能是未知的，因此，使用我们的GPCR小分子化合物库来筛选功能未知的GPCR可能会产生潜在的新型GPCR候选药 ? GPCR化合物库含有与受体相关的小分子， 包括5-HT 受体、多巴胺受体、阿片受体、肾上腺素受体、大麻素受体、mGluR和 ETA-受体等 ? 结构多样，药效显著，可渗透细胞 ? 具有充分详细的结构说明及客户反馈资料 ? NMR和HPLC技术保证产品高纯度 详细信息 配制 1204个化合物预溶于10mM DMSO，80个化合物预溶于10mM水，36个化合物预溶于2mM DMSO，5个化合物预溶于2mM水 容器 带有螺旋盖和二维码的96孔储存管 储存条件 1年 -20°C溶于DMSO 2年 -80°C溶于DMSO Information A unique collection of 1273 small molecules targeting G protein coupled receptors for high throughput screening (HTS) and high content screening (HCS). Description & Advantages ?A unique collection of 1325 small molecules targeting G protein coupled receptors for high throughput screening (HTS) and high content screening (HCS) ? All of the small molecules in the GPCR library are well characterized with biological and pharmaceutical activity ? A powerful tool for discovering GPCR-based drugs that are the richest signal receptor targets for drug discovery ? It is estimated about 200 so-called orphan GPCRs are functionally unknown, as a result, use of our GPCR Small Molecule Compound Library for screening the functionally unknown GPCRs may yield potentially new GPCR-based drug candidates ? The GPCR compound library contains small molecules associated with receptors including 5-HT Receptor, Dopamine Receptor, Opioid Receptor, Adrenergic Receptors, Cannabinoid Receptor, mGluR, and ETA-receptor etc. ? Structurally diverse, medicinally active, and cell permeable ? Rich documentation with structure and customer reviews ? NMR and HPLC validated to ensure the highest purity Product Details Formulation 1204 compounds pre-dissolved in 10mM DMSO, 80 compounds pre-dissolved in 10mM water, 36 compounds pre-dissolved in 2mM DMSO and 5 compounds pre-dissolved in 2mM water Container 96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode Stability 12 months -20°C in DMSO 24 months -80°C in DMSO GPCR Compound Library Composition
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