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TRPM2

Target Id 494
缩写名 SHP2
家族 Transient Receptor Potential channels (TRP)

基因和蛋白信息

Species Transmembrane Domains Amino Acids Chromosomal Location Gene Symbol Gene Name
Human 6 1503 21q22.3 TRPM2 transient receptor potential cation channel subfamily M member 2
Rat 6 1508 20p12 Trpm2 transient receptor potential cation channel, subfamily M, member 2
Mouse 6 1506 10 39.72 cM Trpm2 transient receptor potential cation channel, subfamily M, member 2

作用于该靶标的配体

Ligand Id Ligand Ligand Type Action on Target 对应产品货号 产品名称
2433 2-APB Synthetic organic Antagonist A106408 二苯基硼酸-2-氨基乙酯
2443 ACAA Synthetic organic Antagonist A275778 N-(4-戊基肉桂酰胺)邻氨基苯甲酸(ACA)
2444 ADP ribose Metabolite Agonist A607417 ADP ribose
2391 arachidonic acid Metabolite Potentiation A111764 花生四烯酸(AA)
2445 cADPR Metabolite Agonist C608297 cADPR
2330 clotrimazole Synthetic organic Antagonist C129965 克霉唑
2446 econazole Synthetic organic Antagonist E355746 益康唑
2447 flufenamic acid Synthetic organic Antagonist F129495 氟灭酸
2448 H2O2 Inorganic Agonist H112515 过氧化氢溶液(双氧水)(易制爆)
2449 miconazole Synthetic organic Antagonist M303130 咪康唑
2450 NAADP Metabolite Agonist N348628 烟酸腺嘌呤二核苷酸磷酸钠盐
2451 NAD Metabolite Agonist N432853 β-烟酰胺腺嘌呤二核苷酸 水合物
566 Zn2+ Inorganic None
707 Ca2+ Inorganic None
2346 H+ Inorganic None
4200 GEA 3162 Synthetic organic None G610540 GEA 3162
6333 OAADPR Metabolite Activation O612449 OAADPR
2387 PIP2 Metabolite Activation P612841 PIP?
11080 tatM2NX Peptide Antagonist rp175263 tatM2NX

参考文献

1. Nakayama M, Nakajima D, Nagase T, Nomura N, Seki N, Ohara O.  (1998)  Identification of high-molecular-weight proteins with multiple EGF-like motifs by motif-trap screening..  Genomics,  51  (13):  (27-34).  [PMID:9693030]

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品牌简介

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