TRPM2
Target Id | 494 |
---|---|
缩写名 | SHP2 |
家族 | Transient Receptor Potential channels (TRP) |
基因和蛋白信息
Species | Transmembrane Domains | Amino Acids | Chromosomal Location | Gene Symbol | Gene Name |
---|---|---|---|---|---|
Human | 6 | 1503 | 21q22.3 | TRPM2 | transient receptor potential cation channel subfamily M member 2 |
Rat | 6 | 1508 | 20p12 | Trpm2 | transient receptor potential cation channel, subfamily M, member 2 |
Mouse | 6 | 1506 | 10 39.72 cM | Trpm2 | transient receptor potential cation channel, subfamily M, member 2 |
数据库链接
OMIM | 603749 (Hs) |
---|---|
Entrez Gene | 294329 (Rn) , 28240 (Mm) , 7226 (Hs) |
UniProtKB | Q91YD4 (Mm) , O94759 (Hs) |
RefSeq Protein | NP_003298 (Hs) , NP_001011559 (Rn) , NP_612174 (Mm) |
RefSeq Nucleotide | NM_003307 (Hs) , NM_001011559 (Rn) , NM_138301 (Mm) |
Ensembl Gene | ENSG00000142185 (Hs) , ENSMUSG00000009292 (Mm) , ENSRNOG00000001216 (Rn) |
Protein GI | 58585238 (Rn) , 4507689 (Hs) , 261878536 (Mm) |
ChEMBL Target | CHEMBL1250402 (Hs) |
作用于该靶标的配体
Ligand Id | Ligand | Ligand Type | Action on Target | 对应产品货号 | 产品名称 |
---|---|---|---|---|---|
2433 | 2-APB | Synthetic organic | Antagonist | A106408 | 二苯基硼酸-2-氨基乙酯 |
2443 | ACAA | Synthetic organic | Antagonist | A275778 | N-(4-戊基肉桂酰胺)邻氨基苯甲酸(ACA) |
2444 | ADP ribose | Metabolite | Agonist | A607417 | ADP ribose |
2391 | arachidonic acid | Metabolite | Potentiation | A111764 | 花生四烯酸(AA) |
2445 | cADPR | Metabolite | Agonist | C608297 | cADPR |
2330 | clotrimazole | Synthetic organic | Antagonist | C129965 | 克霉唑 |
2446 | econazole | Synthetic organic | Antagonist | E355746 | 益康唑 |
2447 | flufenamic acid | Synthetic organic | Antagonist | F129495 | 氟灭酸 |
2448 | H2O2 | Inorganic | Agonist | H112515 | 过氧化氢溶液(双氧水)(易制爆) |
2449 | miconazole | Synthetic organic | Antagonist | M303130 | 咪康唑 |
2450 | NAADP | Metabolite | Agonist | N348628 | 烟酸腺嘌呤二核苷酸磷酸钠盐 |
2451 | NAD | Metabolite | Agonist | N432853 | β-烟酰胺腺嘌呤二核苷酸 水合物 |
566 | Zn2+ | Inorganic | None | ||
707 | Ca2+ | Inorganic | None | ||
2346 | H+ | Inorganic | None | ||
4200 | GEA 3162 | Synthetic organic | None | G610540 | GEA 3162 |
6333 | OAADPR | Metabolite | Activation | O612449 | OAADPR |
2387 | PIP2 | Metabolite | Activation | P612841 | PIP? |
11080 | tatM2NX | Peptide | Antagonist | rp175263 | tatM2NX |
参考文献
1. Nakayama M, Nakajima D, Nagase T, Nomura N, Seki N, Ohara O. (1998) Identification of high-molecular-weight proteins with multiple EGF-like motifs by motif-trap screening.. Genomics, 51 (13): (27-34). [PMID:9693030] |