Kir3.4
Target Id | 437 |
---|---|
缩写名 | SHP2 |
家族 | Inwardly rectifying potassium channels (KIR) |
基因和蛋白信息
Species | Transmembrane Domains | Amino Acids | Chromosomal Location | Gene Symbol | Gene Name |
---|---|---|---|---|---|
Human | 2 | 419 | 11q24.3 | KCNJ5 | potassium inwardly rectifying channel subfamily J member 5 |
Rat | 2 | 419 | 8q21 | Kcnj5 | potassium inwardly-rectifying channel, subfamily J, member 5 |
Mouse | 2 | 419 | 9 17.65 cM | Kcnj5 | potassium inwardly-rectifying channel, subfamily J, member 5 |
数据库链接
OMIM | 600734 (Hs) |
---|---|
Entrez Gene | 29713 (Rn) , 16521 (Mm) , 3762 (Hs) |
UniProtKB | P48545 (Mm) , P48548 (Rn) , P48544 (Hs) |
RefSeq Protein | NP_000881 (Hs) , NP_058993 (Rn) , NP_034735 (Mm) |
RefSeq Nucleotide | NM_000890 (Hs) , NM_017297 (Rn) , NM_010605 (Mm) |
Ensembl Gene | ENSG00000120457 (Hs) , ENSMUSG00000032034 (Mm) , ENSRNOG00000033796 (Rn) |
Orphanet | 235181 (Hs) |
Protein GI | 84370254 (Mm) , 24797141 (Hs) , 8393654 (Rn) |
CATH/Gene3D | 2.60.40.1400 (N/A) |
ChEMBL Target | CHEMBL3714708 (Rn) , CHEMBL1914278 (Hs) |
作用于该靶标的配体
Ligand Id | Ligand | Ligand Type | Action on Target | 对应产品货号 | 产品名称 |
---|---|---|---|---|---|
200 | amitriptyline | Synthetic organic | Antagonist | A413377 | 阿米替林 |
2391 | arachidonic acid | Metabolite | Agonist | A111764 | 花生四烯酸(AA) |
2344 | Ba2+ | Inorganic | Antagonist | ||
2398 | clomipramine | Synthetic organic | Antagonist | C608597 | clomipramine |
2356 | Cs+ | Inorganic | Antagonist | ||
2399 | desipramine | Synthetic organic | Antagonist | D609829 | desipramine |
2299 | ethanol | Metabolite | None | E111989 | 乙醇 |
2407 | fingolimod | Synthetic organic | Agonist | F305092 | 芬戈莫德 |
357 | imipramine | Synthetic organic | Antagonist | I611042 | imipramine |
2402 | maprotiline | Synthetic organic | Antagonist | M338146 | 马普替林 |
2340 | Na+ | Inorganic | Agonist | ||
2408 | NIP-142 | Synthetic organic | Antagonist | N335906 | NIP 142 |
2404 | nortriptyline | Synthetic organic | Antagonist | N612368 | nortriptyline |
2341 | phorbol 12-myristate 13-acetate | Synthetic organic | None | P167764 | 佛波醇12-十四酸酯13-乙酸酯 |
2383 | tertiapin-Q | Peptide | Antagonist | rp175271 | tertiapin-Q |
2387 | PIP2 | Metabolite | None | P612841 | PIP? |
7704 | AZD2927 | Synthetic organic | None | A607862 | AZD2927 |
2383 | tertiapin-Q | Peptide | Antagonist | rp175271 | tertiapin-Q |