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Kir3.4

Target Id 437
缩写名 SHP2
家族 Inwardly rectifying potassium channels (KIR)

基因和蛋白信息

Species Transmembrane Domains Amino Acids Chromosomal Location Gene Symbol Gene Name
Human 2 419 11q24.3 KCNJ5 potassium inwardly rectifying channel subfamily J member 5
Rat 2 419 8q21 Kcnj5 potassium inwardly-rectifying channel, subfamily J, member 5
Mouse 2 419 9 17.65 cM Kcnj5 potassium inwardly-rectifying channel, subfamily J, member 5

作用于该靶标的配体

Ligand Id Ligand Ligand Type Action on Target 对应产品货号 产品名称
200 amitriptyline Synthetic organic Antagonist A413377 阿米替林
2391 arachidonic acid Metabolite Agonist A111764 花生四烯酸(AA)
2344 Ba2+ Inorganic Antagonist
2398 clomipramine Synthetic organic Antagonist C608597 clomipramine
2356 Cs+ Inorganic Antagonist
2399 desipramine Synthetic organic Antagonist D609829 desipramine
2299 ethanol Metabolite None E111989 乙醇
2407 fingolimod Synthetic organic Agonist F305092 芬戈莫德
357 imipramine Synthetic organic Antagonist I611042 imipramine
2402 maprotiline Synthetic organic Antagonist M338146 马普替林
2340 Na+ Inorganic Agonist
2408 NIP-142 Synthetic organic Antagonist N335906 NIP 142
2404 nortriptyline Synthetic organic Antagonist N612368 nortriptyline
2341 phorbol 12-myristate 13-acetate Synthetic organic None P167764 佛波醇12-十四酸酯13-乙酸酯
2383 tertiapin-Q Peptide Antagonist rp175271 tertiapin-Q
2387 PIP2 Metabolite None P612841 PIP?
7704 AZD2927 Synthetic organic None A607862 AZD2927
2383 tertiapin-Q Peptide Antagonist rp175271 tertiapin-Q

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品牌简介

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