Kir2.3
Target Id | 432 |
---|---|
缩写名 | SHP2 |
家族 | Inwardly rectifying potassium channels (KIR) |
基因和蛋白信息
Species | Transmembrane Domains | Amino Acids | Chromosomal Location | Gene Symbol | Gene Name |
---|---|---|---|---|---|
Human | 2 | 445 | 22q13.1 | KCNJ4 | potassium inwardly rectifying channel subfamily J member 4 |
Rat | 2 | 446 | 7q34 | Kcnj4 | potassium inwardly-rectifying channel, subfamily J, member 4 |
Mouse | 2 | 445 | 15 37.74 cM | Kcnj4 | potassium inwardly-rectifying channel, subfamily J, member 4 |
数据库链接
OMIM | 600504 (Hs) |
---|---|
Entrez Gene | 116649 (Rn) , 16520 (Mm) , 3761 (Hs) |
UniProtKB | P52189 (Mm) , P52190 (Rn) , P48050 (Hs) |
RefSeq Protein | NP_690607 (Hs) , NP_446322 (Rn) , NP_032453 (Mm) |
RefSeq Nucleotide | NM_152868 (Hs) , NM_053870 (Rn) , NM_008427 (Mm) |
Ensembl Gene | ENSG00000168135 (Hs) , ENSMUSG00000044216 (Mm) , ENSRNOG00000013869 (Rn) |
Protein GI | 158711668 (Mm) , 23110984 (Hs) , 76881824 (Rn) |
CATH/Gene3D | 2.60.40.1400 (N/A) |
ChEMBL Target | CHEMBL2146347 (Hs) |
作用于该靶标的配体
Ligand Id | Ligand | Ligand Type | Action on Target | 对应产品货号 | 产品名称 |
---|---|---|---|---|---|
2391 | arachidonic acid | Metabolite | Agonist | A111764 | 花生四烯酸(AA) |
2344 | Ba2+ | Inorganic | Antagonist | ||
2344 | Ba2+ | Inorganic | Antagonist | ||
2356 | Cs+ | Inorganic | Antagonist | ||
2356 | Cs+ | Inorganic | Antagonist | ||
2346 | H+ | Inorganic | Antagonist | ||
2346 | H+ | Inorganic | Antagonist | ||
708 | Mg2+ | Inorganic | Antagonist | ||
2388 | putrescine | Metabolite | Antagonist | D110948 | (停产)1,4-丁二胺 |
2393 | rose bengal (photoactivated) | Synthetic organic | Antagonist | R613275 | rose bengal (photoactivated) |
943 | SCH-23390 | Synthetic organic | Antagonist | S613487 | SCH-23390 |
2390 | spermidine | Metabolite | Antagonist | S107071 | 亚精胺 |
710 | spermine | Metabolite | Antagonist | ||
2395 | tenidap | Synthetic organic | Agonist | T286898 | Tenidap,环氧合酶(COX-1)抑制剂 |
2343 | tetraethylammonium | Synthetic organic | Antagonist | T614395 | tetraethylammonium |
566 | Zn2+ | Inorganic | Antagonist |