P2Y11 receptor
Target Id | 327 |
---|---|
缩写名 | SHP2 |
家族 | P2Y receptors |
基因和蛋白信息
Species | Transmembrane Domains | Amino Acids | Chromosomal Location | Gene Symbol | Gene Name |
---|---|---|---|---|---|
Human | 7 | 374 | 19p13.2 | P2RY11 | purinergic receptor P2Y11 |
数据库链接
RefSeq Protein | NP_002557 (Hs) |
---|---|
UniProtKB | Q96G91 (Hs) |
OMIM | 602697 (Hs) |
RefSeq Nucleotide | NM_002566 (Hs) |
Entrez Gene | 5032 (Hs) |
Ensembl Gene | ENSG00000244165 (Hs) |
Protein GI | 23463303 (Hs) |
GPCRdb | p2y11_human (Hs) |
Orphanet | 371321 (Hs) |
UniProtKB ID/Entry name | P2Y11_HUMAN (Hs) |
dbSNP | rs3745601 (Hs) |
ChEMBL Target | CHEMBL4867 (Hs) |
作用于该靶标的配体
Ligand Id | Ligand | Ligand Type | Action on Target | 对应产品货号 | 产品名称 |
---|---|---|---|---|---|
1711 | 2MeSATP | Synthetic organic | Full agonist | M607128 | 2MeSATP |
1755 | ADPβS | Synthetic organic | Full agonist | A607416 | ADPβS |
1756 | AR-C67085 | Synthetic organic | Full agonist | A607714 | AR-C67085 |
1713 | ATP | Metabolite | Full agonist | A501266 | 5'-三磷酸腺苷 |
1714 | ATPγS | Synthetic organic | Full agonist | A607804 | ATPγS |
1757 | BzATP | Synthetic organic | Full agonist | B608269 | BzATP |
2450 | NAADP | Metabolite | Full agonist | N348628 | 烟酸腺嘌呤二核苷酸磷酸钠盐 |
2451 | NAD | Metabolite | Full agonist | N432853 | β-烟酰胺腺嘌呤二核苷酸 水合物 |
1734 | UTP | Metabolite | Full agonist | U265870 | (停产)UTP, Molecular Diagnostic Grade sodium salt |
1760 | dATP | Metabolite | Full agonist | D276527 | 2'-脱氧腺苷5'-三磷酸[dATP]三钠三水合物 |
1761 | NF157 | Synthetic organic | Antagonist | N612278 | NF157 |
1762 | NF340 | Synthetic organic | Antagonist | N340885 | NF 340 |
1739 | reactive blue-2 | Synthetic organic | Antagonist | R613114 | reactive blue-2 |
1728 | suramin | Synthetic organic | Antagonist | S614267 | suramin |
4046 | NF546 | Synthetic organic | Full agonist | N288549 | NF 546,P2Y11激动剂 |
1762 | NF340 | Synthetic organic | Antagonist | N340885 | NF 340 |
1712 | ADP | Metabolite | Agonist | A119474 | 腺苷-5’-二磷酸 |
参考文献
1. Hellebrand S, Schaller HC, Wittenberger T. (2000) The brain-specific G-protein coupled receptor GPR85 with identical protein sequence in man and mouse maps to human chromosome 7q31.. Biochim Biophys Acta, 1493 (1-2): (269-72). [PMID:10978537] |