cereblon
Target Id | 3086 |
---|---|
缩写名 | SHP2 |
家族 | E3 ubiquitin ligase components |
基因和蛋白信息
数据库链接
Ensembl Gene | ENSG00000113851 (Hs) , ENSMUSG00000005362 (Mm) , ENSRNOG00000006534 (Rn) |
---|---|
UniProtKB | Q96SW2 (Hs) , Q8C7D2 (Mm) , Q56AP7 (Rn) |
RefSeq Protein | NP_057386 (Hs) , NP_780566 (Mm) , NP_001015003 (Rn) |
Protein GI | 39545580 (Hs) , 28202023 (Mm) , 62543497 (Rn) |
RefSeq Nucleotide | NM_016302 (Hs) , NM_175357 (Mm) , NM_001015003 (Rn) |
OMIM | 609262 (Hs) |
Entrez Gene | 51185 (Hs) , 58799 (Mm) , 297498 (Rn) |
ChEMBL Target | CHEMBL3763008 (Hs) |
作用于该靶标的配体
Ligand Id | Ligand | Ligand Type | Action on Target | 对应产品货号 | 产品名称 |
---|---|---|---|---|---|
7327 | thalidomide | Synthetic organic | Binding | T126856 | (±)-沙利度胺 |
7331 | lenalidomide | Synthetic organic | Binding | L125046 | 来那度胺 |
7348 | pomalidomide | Synthetic organic | Binding | P125813 | 泊马度胺 |
9618 | iberdomide | Synthetic organic | Binding | I414161 | 伊贝多米德(CC220) |
10523 | compound 7f [PMID: 31251063] | Synthetic organic | Binding | N609419 | N-(2,5-Dioxopyrrolidin-3-yl)cinnamamide |
10522 | avadomide | Synthetic organic | Binding | A413866 | Avadomide |
10533 | dTAG-13 | Synthetic organic | Binding | D609997 | dTAG-13 |
10545 | dBRD9 | Synthetic organic | Binding | D609754 | dBRD9 |
11725 | MD-222 | Synthetic organic | Binding | M611763 | MD-222 |
11724 | MG-277 | Synthetic organic | Binding | M611853 | MG-277 |
11799 | SJ995973 | Synthetic organic | Binding | S613596 | SJ995973 |
12000 | MS40 | Synthetic organic | Binding | M612088 | MS40 |
12147 | TL12-186 | Synthetic organic | Binding | T288251 | TL 12-186,多激酶降解PROTAC |
12409 | AK-2292 | Synthetic organic | Binding | A607472 | AK-2292 |
12583 | NVP-DKY709 | Synthetic organic | Binding | N612441 | NVP-DKY709 |