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cereblon

Target Id 3086
缩写名 SHP2
家族 E3 ubiquitin ligase components

基因和蛋白信息

Species Transmembrane Domains Amino Acids Chromosomal Location Gene Symbol Gene Name
Human 2 442 3p26.2 CRBN cereblon
Mouse 2 445 6 E1 Crbn cereblon
Rat 2 445 4q41 Crbn cereblon

作用于该靶标的配体

Ligand Id Ligand Ligand Type Action on Target 对应产品货号 产品名称
7327 thalidomide Synthetic organic Binding T126856 (±)-沙利度胺
7331 lenalidomide Synthetic organic Binding L125046 来那度胺
7348 pomalidomide Synthetic organic Binding P125813 泊马度胺
9618 iberdomide Synthetic organic Binding I414161 伊贝多米德(CC220)
10523 compound 7f [PMID: 31251063] Synthetic organic Binding N609419 N-(2,5-Dioxopyrrolidin-3-yl)cinnamamide
10522 avadomide Synthetic organic Binding A413866 Avadomide
10533 dTAG-13 Synthetic organic Binding D609997 dTAG-13
10545 dBRD9 Synthetic organic Binding D609754 dBRD9
11725 MD-222 Synthetic organic Binding M611763 MD-222
11724 MG-277 Synthetic organic Binding M611853 MG-277
11799 SJ995973 Synthetic organic Binding S613596 SJ995973
12000 MS40 Synthetic organic Binding M612088 MS40
12147 TL12-186 Synthetic organic Binding T288251 TL 12-186,多激酶降解PROTAC
12409 AK-2292 Synthetic organic Binding A607472 AK-2292
12583 NVP-DKY709 Synthetic organic Binding N612441 NVP-DKY709

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品牌简介

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