carbonic anhydrase 12
Target Id | 2747 |
---|---|
缩写名 | CA XII |
家族 | Carbonic anhydrases |
基因和蛋白信息
数据库链接
RefSeq Nucleotide | NM_013040 (Rn) , NM_178396 (Mm) , NM_001218 (Hs) |
---|---|
RefSeq Protein | NP_037172 (Rn) , NP_848483 (Mm) , NP_001209 (Hs) |
Ensembl Gene | ENSRNOG00000017766 (Rn) , ENSMUSG00000032373 (Mm) , ENSG00000074410 (Hs) |
OMIM | 603263 (Hs) |
UniProtKB | O43570 (Hs) , Q8CI85 (Mm) |
Protein GI | 4502515 (Hs) , 227496587 (Mm) , 19923678 (Rn) |
CATH/Gene3D | 3.10.200.10 (N/A) |
ChEMBL Target | CHEMBL3242 (Hs) |
作用于该靶标的配体
Ligand Id | Ligand | Ligand Type | Action on Target | 对应产品货号 | 产品名称 |
---|---|---|---|---|---|
6792 | acetazolamide | Synthetic organic | Inhibition | A194116 | 乙酰唑胺 |
6807 | diclofenamide | Synthetic organic | Inhibition | D129876 | 双氯非那胺 |
6814 | ethoxzolamide | Synthetic organic | Inhibition | E300261 | 6-乙氧基-2-苯并噻唑苯磺酸 |
6828 | methazolamide | Synthetic organic | Inhibition | M303972 | 醋甲唑胺 |
6810 | dorzolamide | Synthetic organic | Inhibition | D349665 | 多佐胺 |
6797 | brinzolamide | Synthetic organic | Inhibition | B129826 | 布林佐胺 |
6849 | topiramate | Synthetic organic | Inhibition | T115813 | 托吡酯 |
6920 | benzolamide | Synthetic organic | Inhibition | B607993 | benzolamide |
5501 | sulpiride | Synthetic organic | Inhibition | P160775 | (±)-舒必利 |
2892 | celecoxib | Synthetic organic | Inhibition | C129279 | 塞来昔布 |
2894 | valdecoxib | Synthetic organic | Inhibition | V125795 | 代他考昔 |
7046 | indisulam | Synthetic organic | Inhibition | I305112 | Indisulam,分子胶 |
7047 | zonisamide | Synthetic organic | Inhibition | Z163001 | 唑尼沙胺 |
7147 | chlorthalidone | Synthetic organic | Inhibition | C304602 | 氯塞酮 |
10149 | SLC-0111 | Synthetic organic | Inhibition | U129821 | U-104,碳酸酐酶(CA)IX和XII抑制剂 |
10433 | compound 5a [PMID: 31287314] | Synthetic organic | Inhibition | P609318 | 4-(prop-2-ynylamino)benzenesulfonamide |
10434 | compound 5b [PMID: 31287314] | Synthetic organic | Inhibition | C609324 | compound 5b |