proteasome 20S subunit beta 5
Target Id | 2406 |
---|---|
缩写名 | SHP2 |
家族 | T1: Proteasome |
基因和蛋白信息
数据库链接
OMIM | 600306 (Hs) |
---|---|
Entrez Gene | 5693 (Hs) , 19173 (Mm) , 29425 (Rn) |
UniProtKB | P28074 (Hs) , O55234 (Mm) , P28075 (Rn) |
RefSeq Protein | NP_001124197 (Hs) , NP_001138404 (Hs) , NP_002788 (Hs) , NP_035316 (Mm) , NP_001099197 (Rn) |
RefSeq Nucleotide | NM_001130725 (Hs) , NM_001144932 (Hs) , NM_002797 (Hs) , NM_011186 (Mm) , NM_001105727 (Rn) |
Ensembl Gene | ENSG00000100804 (Hs) , ENSMUSG00000022193 (Mm) , ENSRNOG00000013386 (Rn) |
MEROPS | T01.P01 (Hs) |
Protein GI | 195539356 (Hs) , 222144262 (Hs) , 4506201 (Hs) , 6755204 (Mm) , 160333293 (Rn) |
DrugBank Target | P28074 (Hs) |
CATH/Gene3D | 3.60.20.10 (N/A) |
ChEMBL Target | CHEMBL4662 (Hs) , CHEMBL4523208 (Rn) , CHEMBL1944494 (Mm) |
作用于该靶标的配体
Ligand Id | Ligand | Ligand Type | Action on Target | 对应产品货号 | 产品名称 |
---|---|---|---|---|---|
6391 | bortezomib | Synthetic organic | Inhibition | B125789 | TCN 213,可逆蛋白酶体抑制剂 |
8450 | ixazomib | Synthetic organic | Inhibition | M128010 | 伊沙佐米(MLN2238) |
8616 | MG-132 | Peptide | Inhibition | M276573 | MG-132(乙醇溶液) |
8618 | compound 3b [PMID: 24946214] | Synthetic organic | Inhibition | R609166 | [(1R)-3-methyl-1-[3-(1-oxoisoquinolin-2-yl)propanoylamino]butyl]boronic acid |
8739 | oprozomib | Synthetic organic | Inhibition | O129260 | Oprozomib (ONX 0912),抑制20S蛋白酶体β5/LMP7的CT-L活性 |
7420 | carfilzomib | Synthetic organic | Inhibition | C127870 | 卡非佐米 |
10409 | KZR-616 | Synthetic organic | Inhibition | K611367 | KZR-616 |
11321 | WLL-vs | Synthetic organic | Inhibition | W614850 | WLL-vs |
12174 | NIC-0102 | Synthetic organic | Inhibition | R612294 | [(1R)-1-[[(2S)-2-[(2,6-difluorobenzoyl)amino]-3-phenylpropanoyl]amino]-3-methylbutyl]boronic acid |