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proteasome 20S subunit beta 5

Target Id 2406
缩写名 SHP2
家族 T1: Proteasome

基因和蛋白信息

Species Transmembrane Domains Amino Acids Chromosomal Location Gene Symbol Gene Name
Human 2 263 14q11.2 PSMB5 proteasome 20S subunit beta 5
Mouse 2 264 14 27.86 cM Psmb5 proteasome (prosome, macropain) subunit, beta type 5
Rat 2 263 15p13 Psmb5 proteasome 20S subunit beta 5

作用于该靶标的配体

Ligand Id Ligand Ligand Type Action on Target 对应产品货号 产品名称
6391 bortezomib Synthetic organic Inhibition B125789 TCN 213,可逆蛋白酶体抑制剂
8450 ixazomib Synthetic organic Inhibition M128010 伊沙佐米(MLN2238)
8616 MG-132 Peptide Inhibition M276573 MG-132(乙醇溶液)
8618 compound 3b [PMID: 24946214] Synthetic organic Inhibition R609166 [(1R)-3-methyl-1-[3-(1-oxoisoquinolin-2-yl)propanoylamino]butyl]boronic acid
8739 oprozomib Synthetic organic Inhibition O129260 Oprozomib (ONX 0912),抑制20S蛋白酶体β5/LMP7的CT-L活性
7420 carfilzomib Synthetic organic Inhibition C127870 卡非佐米
10409 KZR-616 Synthetic organic Inhibition K611367 KZR-616
11321 WLL-vs Synthetic organic Inhibition W614850 WLL-vs
12174 NIC-0102 Synthetic organic Inhibition R612294 [(1R)-1-[[(2S)-2-[(2,6-difluorobenzoyl)amino]-3-phenylpropanoyl]amino]-3-methylbutyl]boronic acid

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品牌简介

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