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GPR119

Target Id 126
缩写名 SHP2
家族 GPR18, GPR55 and GPR119

基因和蛋白信息

Species Transmembrane Domains Amino Acids Chromosomal Location Gene Symbol Gene Name
Rat 7 468 Xq36 Gpr119 G protein-coupled receptor 119
Human 7 335 Xq26.1 GPR119 G protein-coupled receptor 119
Mouse 7 335 X A5 Gpr119 G-protein coupled receptor 119

作用于该靶标的配体

Ligand Id Ligand Ligand Type Action on Target 对应产品货号 产品名称
3318 PSN375963 Synthetic organic Agonist P347546 PSN 375963盐酸盐
3319 PSN632408 Synthetic organic Agonist P612998 PSN632408
4027 AS1269574 Synthetic organic Agonist A288879 AS 1269574,GPR119受体激动剂
2661 N-oleoylethanolamide Metabolite Agonist Z130746 油酰单乙醇胺
3622 N-palmitoylethanolamine Metabolite Full agonist N135851 十六酰胺乙醇
3621 SEA Metabolite Full agonist S351349 硬脂酰乙醇酰胺
3623 oleoyl-lysophosphatidylcholine Synthetic organic Agonist O130376 1-油酰基-2-羟基-sn-甘油-3-磷酸胆碱
5650 1-palmitoyl-lysophosphatidylcholine Metabolite Agonist P130493 1-棕榈酰-sn-甘油-3-磷酸胆碱
5651 1-stearoyl-lysophosphatidylcholine Metabolite Agonist S130495 1-硬脂酰-sn-甘油-3-磷酰胆碱
4028 lysophosphatidylinositol Metabolite Agonist L611690 lysophosphatidylinositol
5652 lysophosphatidylethanolamine Metabolite Agonist L611689 lysophosphatidylethanolamine
5653 AR231453 Synthetic organic Agonist A275017 AR 231453,GPR119激动剂
2488 olvanil Synthetic organic Agonist O286933 Olvanil,TRPV激动剂 (顺反异构体混合物)
5552 N-oleoyldopamine Metabolite Agonist O287241 OLDA,内源性TRPV1激动剂
5720 (R)-N-oleoyltyrosinol Synthetic organic Agonist R613225 (R)-N-oleoyltyrosinol
5721 (S)-N-oleoyltyrosinol Synthetic organic Agonist O340917 OMDM-1
5722 AS1535907 Synthetic organic Agonist A607752 AS1535907
5723 AS1907417 Synthetic organic Agonist A607755 AS1907417
5112 2-oleoyl glycerol Metabolite Agonist
5724 compound 3 [PMID: 21310611] Synthetic organic Agonist M609190 (1-methylcyclopropyl) 4-[(1S)-1-fluoro-2-[[2-(2,3,6-trifluorophenyl)acetyl]amino]ethyl]piperidine-1-carboxylate
5727 JNJ-38431055 Synthetic organic Agonist A412183 APD597
5735 compound 42 [PMID: 22545772] Synthetic organic Agonist S609226 4-[({2-[(2S)-2-methyl-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazin-1-yl]pyrimidin-5-yl}oxy)methyl]pyridine-3-carbonitrile
5737 compound 3a [PMID: 21444206] Synthetic organic Agonist T609163 tert-butyl 4-[1-(4-methylsulfonylphenyl)pyrazolo[4,5-e]pyrimidin-4-yl]oxypiperidine-1-carboxylate
5738 compound 3j [PMID: 21444206] Synthetic organic Agonist T609175 tert-butyl 4-{[1-(2-fluoro-4-methanesulfonylphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]oxy}piperidine-1-carboxylate
5739 compound 8g [PMID: 21444206] Synthetic organic Agonist T609458 tert-butyl 4-{[1-(2-fluoro-4-methanesulfonylphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]sulfanyl}piperidine-1-carboxylate
5740 compound 23 [PMID: 21444206] Synthetic organic Agonist T608971 tert-butyl 4-{[9-(2-fluoro-4-methanesulfonylphenyl)-8-oxo-8,9-dihydro-7H-purin-6-yl]oxy}piperidine-1-carboxylate
5741 compound 29a [PMID: 21444206] Synthetic organic Agonist T609038 tert-butyl 4-[[3-(4-methylsulfonylphenyl)-[1,2]oxazolo[5,4-e]pyrimidin-7-yl]oxy]piperidine-1-carboxylate
5743 compound 1 [PMID: 21939274] Synthetic organic Agonist P608880 propan-2-yl 4-[3-cyano-5-(quinoxalin-6-yl)pyridin-2-yl]piperazine-1-carboxylate
5744 compound 2 [PMID: 21939274] Synthetic organic Agonist C609078 5-(4-cyano-3-methylphenyl)-2-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyridine-3-carbonitrile
5745 compound 1 [PMID: 21273063] Synthetic organic Agonist T608877 tert-butyl 4-[1-(pyridin-3-yl)piperidin-4-yl]piperidine-1-carboxylate
5747 compound 36 [PMID: 21273063] Synthetic organic Agonist E609138 2-ethynyl-4-methyl-6-{4-[1-(5-methylpyrazin-2-yl)piperidin-4-yl]piperidin-1-yl}pyrimidine
5748 compound 58 [PMID: 21273063] Synthetic organic Agonist C609311 5-chloro-2-{4-[(1R,2S)-2-{2-[(5-methanesulfonylpyridin-2-yl)oxy]ethyl}cyclopropyl]piperidin-1-yl}pyrimidine
5755 compound 36j [PMID: 21536438] Synthetic organic Agonist C609136 3-chloro-4-[(6-{[(1S,5S)-8-(cyclopropanesulfonyl)-8-azabicyclo[3.2.1]octan-3-yl]oxy}-5-methylpyrimidin-4-yl)amino]benzonitrile
5750 compound 20f [PMID: 21536438] Synthetic organic Agonist T608911 tert-butyl (1S,5S)-3-({5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}oxy)-8-azabicyclo[3.2.1]octane-8-carboxylate
5756 1-oleoyl glycerol Synthetic organic Agonist M107453 甘油单油酸酯
10082 DS-8500a Synthetic organic Agonist D609984 DS-8500a
10137 YH18968 Synthetic organic Agonist Y614911 YH18968
10166 MBX-2982 Synthetic organic Agonist M127623 MBX-2982
12151 APD668 Synthetic organic Agonist A413612 APD668
12151 APD668 Synthetic organic Agonist A413612 APD668

参考文献

1. Pérez Jurado LA, Li X, Francke U.  (1995)  The human calcitonin receptor gene (CALCR) at 7q21.3 is outside the deletion associated with the Williams syndrome..  Cytogenet Cell Genet,  70  (3-4):  (246-9).  [PMID:7789182]

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品牌简介

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